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Total synthesis of derivatives of (±)-6-oxa and aza-estrone

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Zusammenfassung

Es wird über die Totalsynthese von verschiedenen Derivaten des (±)-6-Oxa- und Aza-Östrons und die Umwandlung von (±)-17β-Oxy-3-methoxy-6-oxa-östratrien-1, 3, 510 zu Verbindungen der (±)-19-Nor-6-oxa-testosteron-Klasse berichtet. Die biologische Wirksamkeit der Glieder in der 6-Oxa-Reihe wird beschrieben.

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Literatur

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Authors and Affiliations

  1. Research Division, Wyeth Laboratories Inc., Philadelphia, Pennsylvania, USA

    H. Smith, G. H. Douglas & C. R. Walk

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  1. H. Smith
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  2. G. H. Douglas
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  3. C. R. Walk
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Smith, H., Douglas, G.H. & Walk, C.R. Total synthesis of derivatives of (±)-6-oxa and aza-estrone. Experientia 20, 418–419 (1964). https://doi.org/10.1007/BF02152119

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