Elsevier

Tetrahedron Letters

Volume 40, Issue 35, 27 August 1999, Pages 6493-6496
Tetrahedron Letters

A convenient one-pot synthesis of N-aryl-3-pyrrolines

https://doi.org/10.1016/S0040-4039(99)01334-9Get rights and content

Abstract

N-propargylanilines, under one-pot homologation conditions, undergo an in situ cyclisation catalysed by Cu(I) to yield 3-pyrrolines in good yield.

N-propargylanilines under one-pot homologation conditions undergo an in situ cyclisation catalysed by Cu(I) to yield 3-pyrrolines in good yield.

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