Synthesis of Functionalized Indoles by Diels-Alder Reaction Utilizing the Diene Generated by the Alkylation of N-Methyl-3-thioacetylpyrrole

Masayuki MURASE; Shinya YOSHIDA; Toshihiro HOSAKA; Seisho TOBINAGA

doi:10.1248/cpb.39.489

Masayuki MURASE, Shinya YOSHIDA, Toshihiro HOSAKA, Seisho TOBINAGA

Author information

Keywords: cycloaddition, 3-vinylpyrrole, 1-methyl-3-thioacetylpyrrole, alkylation, dienophile, indole

JOURNAL FREE ACCESS

1991 Volume 39 Issue 2 Pages 489-492

DOI https://doi.org/10.1248/cpb.39.489

Details

Abstract

Cycloaddition reaction of 3-vinylpyrroles, generated by the alkylation of 1-methyl-3-thioacetylpyrrole, with dienophiles provided functionalized indoles.

Corresponding author

Register with J-STAGE for free!